O antagonista do receptor de neuroquinina-1 aprepitante diminui a eficácia da quimioterapia baseada em ciclofosfamida?

Autores

  • Carlos Eduardo Paiva
  • Bianca Sakamoto Ribeiro Paiva
  • Odair Carlito Michelin

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Biografia do Autor

Carlos Eduardo Paiva

MD, MSc. PhD student and clinical oncologist, Oncological and Hemato-Oncological Center, Universidade Estadual Paulista (Unesp), Botucatu, São Paulo, Brazil.

Bianca Sakamoto Ribeiro Paiva

RN, MSc. PhD student and assistant nursing professor, Department of Nursing, Botucatu Medical School, Universidade Estadual Paulista (Unesp), Botucatu, São Paulo, Brazil.

Odair Carlito Michelin

MD, PhD. Associate professor, Department of Clinics, Botucatu Medical School, Universidade Estadual Paulista (Unesp), Botucatu, São Paulo, Brazil.

Referências

Warr DG, Grunberg SM, Gralla RJ, et al. The oral NK(1) antagonist aprepitant for the preven- tion of acute and delayed chemotherapy-induced nausea and vomiting: Pooled data from 2 randomised, double-blind, placebo controlled trials. Eur J Cancer. 2005;41(9):1278-85.

Warr DG, Hesketh PJ, Gralla RJ, et al. Efficacy and tolerability of aprepitant for the prevention of chemotherapy-induced nausea and vomiting in patients with breast cancer after mode- rately emetogenic chemotherapy. J Clin Oncol. 2005;23(12):2822-30.

van Schaik RH. CYP450 pharmacogenetics for personalizing cancer therapy. Drug Resist Updat. 2008;11(3):77-98.

de Jonge ME, Huitema AD, Holtkamp MJ, van Dam SM, Beijnen JH, Rodenhuis S. Aprepi- tant inhibits cyclophosphamide bioactivation and thiotepa metabolism. Cancer Chemother Pharmacol. 2005;56(4):370-8.

Yeo W, Mo FK, Suen JJ, et al. A randomized study of aprepitant, ondansetron and dexametha- sone for chemotherapy-induced nausea and vomiting in Chinese breast cancer patients recei- ving moderately emetogenic chemotherapy. Breast Cancer Res Treat. 2009;113(3):529-35.

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Publicado

2009-11-11

Como Citar

1.
Paiva CE, Paiva BSR, Michelin OC. O antagonista do receptor de neuroquinina-1 aprepitante diminui a eficácia da quimioterapia baseada em ciclofosfamida?. Sao Paulo Med J [Internet]. 11º de novembro de 2009 [citado 10º de março de 2025];127(6):385-6. Disponível em: https://periodicosapm.emnuvens.com.br/spmj/article/view/1927

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